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Kappa agonists, Opioid receptor ligands, Drugs acting on the nervous system, Allyl compounds, Six-membered rings, Alkenes

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Analgesics (1)
Cyclic compounds (1)
Cycloalkenes (1)
Cyclohexenes (1)
Dissociative drugs (1)
Opioid antagonists (1)
Opioids (1)
Pharmaceuticals (1)
Psychoactive drugs (1)
Semisynthetic opioids (1)

Nalorphine (62-67-9)  
Allylnormorphine  ·  Nalorphine Hydrochloride  ·  Lethidrone
Nalorphine (INN) (brand names Lethidrone, Nalline), also known as N-allylnormorphine, is a mixed opioid agonist–antagonist with opioid antagonist and analgesic properties. It was introduced in 1954 and was used as an antidote to reverse opioid overdose and in a challenge test to determine opioid dependence. It acts at two opioid receptors — the μ-opioid receptor (MOR) where it has antagonistic effects, and at the κ-opioid receptor (KOR) (Ki = 1.6 nM; EC50 = 483 nM; Emax = 95%) where it exerts high-efficacy partial agonist/near-full agonist characteristics.

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TENOCYCLIDINE (21500-98-1, 1867-65-8)  
Tenocyclidine (TCP) was discovered by a team at Parke Davis in the late 1950s. It is a dissociative anesthetic drug with psychostimulant and hallucinogenic effects. It is similar in effects to phencyclidine (PCP) but is considerably more potent.
2-Hydroxybenzophenone (117-99-7)  
ortho-hydroxybenzophenone
1,3-Bis(4-piperidyl)propane (16898-52-5)  
1,3-bis(4-piperidinyl)propane
4-Hydroxybenzophenone (1137-42-4)  
4-hydroxybenzophenone, ion(1-)  ·  para-hydroxybenzophenone
Indoline (496-15-1)  
2,3-dihydro-1H-indole
Indoline is an aromatic heterocyclic organic compound with the chemical formula C8H9N. It has a bicyclic structure, consisting of a six-membered benzene ring fused to a five-membered nitrogen-containing ring. The compound is based on the indole structure, but the 2-3 bond is saturated.
PIPERIDINE (110-89-4)  
Piperidine is an organic compound with the molecular formula (CH2)5NH. This heterocyclic amine consists of a six-membered ring containing five methylene bridges (–CH2–) and one amine bridge (–NH–). It is a colorless liquid with an odor described as objectionable, and typical of amines.
Azacyclonol (115-46-8)  
azacyclonol hydrochloride
Azacyclonol (trade names Ataractan, Calmeran, Frenoton, Frenquel, Psychosan), also known as γ-pipradrol, is a drug which is an ataractive; an agent which diminishes hallucinations in psychotic individuals. It has also been called a tranquilizer and antipsychotic, though these definitions are not accurate as it does not actually possess such properties. Despite being a positional isomer of pipradrol, it is not a psychostimulant, and instead has mild depressant effects.
Related searches
Kappa agonists
Opioid receptor ligands
Drugs acting on the nervous system
Allyl compounds
Six-membered rings
Alkenes
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