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Kappa agonists, Opioid receptor ligands, Drugs acting on the nervous system, Tetrahydrofurans

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Analgesics (3)
Cyclic compounds (3)
Five-membered rings (3)
Opioids (3)
Psychoactive drugs (3)
Pyrrolidines (3)
Spiro compounds (3)
Dissociative drugs (2)
Psychedelic drugs (2)
Psychoactive drug (2)
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ENADOLINE (124378-77-4)  
Enadoline is a drug which acts as a highly selective κ-opioid agonist. In human studies, it produced visual distortions and feelings of dissociation, reminiscent of the effects of salvinorin A. It was studied as a potential analgesic, but abandoned because of the dose-limiting effects of dysphoria, which could be expected from a κ-opioid agonist.
U-69593 (96744-75-1)  
U-69,593 is a drug which acts as a potent and selective κ1-opioid receptor agonist. In animal studies it has been shown to produce antinociception, anti-inflammation, anxiolysis (at low doses), respiratory depression, and diuresis, while having little effect on gastrointestinal motility. It also inhibits the peripheral, though not central secretion of oxytocin and vasopressin in rats.
Related searches
Kappa agonists
Opioid receptor ligands
Drugs acting on the nervous system
Tetrahydrofurans