Kappa agonists, Opioid receptor ligands, Drugs acting on the nervous system, Thiophenes, Opioids, Benzodiazepines
Cyclic compounds (1)
KC 5103 · KC 5911 · KC-5911
Tifluadom is a benzodiazepine derivative with an unusual activity profile. Unlike most benzodiazepines, tifluadom has no activity at the GABAA receptor, but instead is a selective agonist for the κ-opioid receptor. In accordance, it has potent analgesic and diuretic effects in animals, and also has sedative effects and stimulates appetite.