877-202-0205     support@chemchart.com     @chemchart
        
Sign In    Register
   Reset Filters

Pyrazoles, Opioids, Iodoarenes

Categories

AM cannabinoids (1)
Analgesics (1)
Aromatic compounds (1)
Cannabinoid (1)
Cannabinoids (1)
Cannabis (1)
Chloroarenes (1)
Cyclic compounds (1)
Drugs acting on the nervous system (1)
Five-membered rings (1)
Opioid antagonists (1)
Opioid receptor ligands (1)
Piperidines (1)
Psychoactive drug (1)
Psychoactive drugs (1)
Pyrazolecarboxamides (1)
Six-membered rings (1)

Suppliers

Sigma Aldrich (1)

AM251 (183232-66-8)  
AM 251  ·  N-(piperidin-1-yl)-1-(2,4-dichlorophenyl)-5-(4-iodophenyl)-4-methyl-1H-pyrazole-3-carboxamide  ·  N-(piperidin-1-yl)-5-(4-iodophenyl)-1-(2,4-dichlorophenyl)-4-methyl-1H-pyrazole-3-carboxamide
AM-251 is an inverse agonist at the CB1 cannabinoid receptor. AM-251 is structurally very close to SR141716A (rimonabant); both are biarylpyrazole cannabinoid receptor antagonists. In AM-251 the p-chloro group attached to the phenyl substituent at C-5 of the pyrazole ring is replaced with a p-iodo group.
Related searches
Pyrazoles
Opioids
Iodoarenes